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Pepstatin (Trifluoroacetate)

Pepstatin (Trifluoroacetate)

€31.00

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Item no.	HY-P0018A-5mg
Manufacturer	MedChem Express
Amount	5 mg
Category	Reagents & Chemicals Other Chemicals
Type	Chemicals
Specific against	other
Purity	98.77
Formula	C36H64F3N5O11
Citations	Int J Antimicrob Agents. 2019 Dec;54(6):814-819. Adv Sci (Weinh). 2022 Oct 10;e2203831. Arch Biochem Biophys. 2023 May 22, 109646. Biochem Bioph Res Co. 2020 Sep 10;530(1):292-300. Cancer Lett. 2022 Mar 9;215629. Carbohydr Polym. 2023 Jul 17, 121208. Cell Death Dis. 2022 Dec 16;13(12):1048. Cell Rep. 2021 Nov 2;37(5):109931. Environ Sci Technol. 2017 Dec 5;51(23):13938-13948. Eur J Pharmacol. 2022 Feb 11;920:174823. FASEB J. 2022 Jan;36(1):e22121. Int J Oncol. 2019 Jul;55(1):331-339. J Virol. 2021 Sep 22;JVI0153721. J Virol. 2023 Oct 17:e0107523. Mol Med Rep. 2019 Jan;19(1):41-50. Pharmaceuticals. 2022, 15(12), 1509 Pharmacol Res. 2021 Dec 1;175:105985. Sci Adv. 2022 Nov 11;8(45):eabn6579. SSRN. 2023 Apr 10. Toxicol Appl Pharmacol. 2018 Oct 1;356:159-171. Biol Pharm Bull. 2022 Feb 3. [1]Umezawa H, et al. Pepstatin, a new pepsin inhibitor produced by Actinomycetes. J Antibiot (Tokyo). 1970 May;23(5):259-62. [2]Seelmeier S, et al. Human immunodeficiency virus has an aspartic-type protease that can be inhibited by pepstatin A. Proc Natl Acad Sci U S A. 1988 Sep;85(18):6612-6.
Smiles	OC(C(F)(F)F)=O.CC(C[C@H](NC([C@@H](NC([C@@H](NC(CC(C)C)=O)C(C)C)=O)C(C)C)=O)[C@@H](O)CC(N[C@@H](C)C(N[C@@H](CC(C)C)[C@@H](O)CC(O)=O)=O)=O)C
ECLASS 10.1	32160000
ECLASS 11.0	32160000
UNSPSC	12000000
Alias	Pepstatin A (Trifluoroacetate)
Available
Product Description	Pepstatin (Pepstatin A) Trifluoroacetate is a specific, orally active aspartic protease inhibitor produced by actinomycetes, with IC50s of 4.5 nM, 6.2 nM, 150 nM, 290 nM, 520 nM and 260 nM for hemoglobin-pepsin, hemoglobin-proctase, casein-pepsin, casein-proctase, casein-acid protease and hemoglobin-acid protease, respectively. Pepstatin Trifluoroacetate also inhibits HIV protease[1][2].
StorageTemperature	-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Shipping	Blue Ice
Manufacturers Applications	COVID-19-anti-virus
Molecular Weight	799.92
Clinical Information	No Development Reported
Solubility	DMSO : 100 mg/mL (ultrasonic)
Pathway	Anti-infection; Autophagy; Metabolic Enzyme/Protease
Manufacturers Product type	Peptides

Note: The presented information and documents (Manual, Product Datasheet, Safety Datasheet and Certificate of Analysis) correspond to our latest update and should serve for orientational purpose only. We do not guarantee the topicality. We would kindly ask you to make a request for specific requirements, if necessary.

All products are intended for research use only (RUO). Not for human, veterinary or therapeutic use.

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Amount: 5 mg

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